α-Conotoxin PIA
CAS No. 669050-68-4
α-Conotoxin PIA ( )
Catalog No. M30729 CAS No. 669050-68-4
Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM for rat α6/α3β2β3 and α3β2 receptors respectively).
Purity : >98% (HPLC)
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Biological Information
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Product Nameα-Conotoxin PIA
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NoteResearch use only, not for human use.
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Brief DescriptionSelective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM for rat α6/α3β2β3 and α3β2 receptors respectively).
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DescriptionSelective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM for rat α6/α3β2β3 and α3β2 receptors respectively).
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Synonyms
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PathwayEndocrinology/Hormones
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TargetAChR
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number669050-68-4
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Formula Weight1981.3
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Molecular FormulaC79H125N27O25S4
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Purity>98% (HPLC)
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Solubilitywater:2 mg/mL
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SMILES[H]N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(O)=O)C(=O)N1CCC[C@H]1C(=O)N[C@H]1CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@@H]3CCCN3C(=O)[C@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CSSC[C@H](NC(=O)C(NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]3CCCN3C(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC3=CNC=N3)NC(=O)[C@@H](NC(=O)C(NC2=O)[C@@H](C)O)C(C)C)[C@@H](C)CC)C(N)=O)NC1=O)C(C)C
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Chemical Name
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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2,3-Dihydrobenzofura...
2,3-Dihydrobenzofuran is an acetylcholinesterase (AChE) inhibitor isolated from leaves of L. camara.?Coumaran can be used as a biopesticide.?2,3-dihydrobenzofuran is a member of the class of 1-benzofurans that is the 2,3-dihydroderivative of benzofuran.?It has a role as a metabolite.The in vitro inhibition of acetylcholinesterase was increased with the concentration of Coumaran in the housefly (head and thorax) homogenate.
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Anisotropine Methylb...
Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.
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Dichlorisone Acetate
It belongs to organophosphate compounds, used as a kind of common environmental health insecticide.